2. GPCR/G Protein
  3. Adenosine Receptor
  4. MRS-3777 hemioxalate

MRS-3777 hemioxalate 

Cat. No.: HY-110037 Purity: 95.64%
COA Handling Instructions

MRS-3777 hemioxalate is a selective adenosine A3 receptor antagonist.

For research use only. We do not sell to patients.

MRS-3777 hemioxalate Chemical Structure

MRS-3777 hemioxalate Chemical Structure

CAS No. : 1186195-57-2

Size Price Stock Quantity
Solution
10 mM * 1 mL in DMSO USD 132 In-stock
Solid + Solvent
10 mM * 1 mL
ready for reconstitution
 USD 132 In-stock
Solid
5 mg USD 120 In-stock
10 mg USD 200 In-stock
25 mg USD 400 In-stock
50 mg USD 650 In-stock
100 mg   Get quote  
200 mg   Get quote  

* Please select Quantity before adding items.

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Based on 1 publication(s) in Google Scholar

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Adenosine A1 receptor (A1R) Adenosine A2A receptor (A2AR) Adenosine A2B receptor (A2BR) Adenosine A3 receptor (A3R)

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  • Purity & Documentation

  • References

  • Customer Review

Description

MRS-3777 hemioxalate is a selective adenosine A3 receptor antagonist[1].

IC50 & Target

adenosine A3 receptor[1]
Molecular Weight

399.40

Appearance

Solid

Formula

C17H19N5O.1/2C2H2O4
CAS No.
SMILES

OC(C(O)=O)=O.C1(NC2CCCCC2)=C3C(N=CN3)=NC(OC4=CC=CC=C4)=N1.[1/2]
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

-20°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (250.38 mM; ultrasonic and adjust pH to 3 with HCl)

H2O : < 0.1 mg/mL (insoluble)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.5038 mL 12.5188 mL 25.0376 mL
5 mM 0.5008 mL 2.5038 mL 5.0075 mL
10 mM 0.2504 mL 1.2519 mL 2.5038 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: 2.5 mg/mL (6.26 mM); Suspended solution; Need ultrasonic

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: 2.5 mg/mL (6.26 mM); Suspended solution; Need ultrasonic

  • 3.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.5 mg/mL (6.26 mM); Clear solution

*All of the co-solvents are available by MCE.
Purity & Documentation
References
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

MRS-3777 hemioxalate1186195-57-2Adenosine ReceptorP1 receptorInhibitorinhibitorinhibit

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