1. GPCR/G Protein
  2. Adenosine Receptor
  3. MRS-3777 hemioxalate

MRS-3777 hemioxalate 

Cat. No.: HY-110037 Purity: 95.64%
Handling Instructions

MRS-3777 hemioxalate is a selective adenosine A3 receptor antagonist.

For research use only. We do not sell to patients.

MRS-3777 hemioxalate Chemical Structure

MRS-3777 hemioxalate Chemical Structure

CAS No. : 1186195-57-2

Size Price Stock Quantity
Solution
10 mM * 1 mL in DMSO USD 132 In-stock
Estimated Time of Arrival: December 31
Solid + Solvent
10 mM * 1 mL
ready for reconstitution
USD 132 In-stock
Estimated Time of Arrival: December 31
Solid
5 mg USD 120 In-stock
Estimated Time of Arrival: December 31
10 mg USD 200 In-stock
Estimated Time of Arrival: December 31
25 mg USD 400 In-stock
Estimated Time of Arrival: December 31
50 mg USD 650 In-stock
Estimated Time of Arrival: December 31
100 mg   Get quote  
200 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

Based on 1 publication(s) in Google Scholar

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Description

MRS-3777 hemioxalate is a selective adenosine A3 receptor antagonist[1].

IC50 & Target

adenosine A3 receptor[1]

Molecular Weight

399.40

Formula

C₁₇H₁₉N₅O.₁/₂C₂H₂O₄

CAS No.
SMILES

OC(C(O)=O)=O.C1(NC2CCCCC2)=C3C(N=CN3)=NC(OC4=CC=CC=C4)=N1.[1/2]

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (250.38 mM; ultrasonic and adjust pH to 3 with HCl)

H2O : < 0.1 mg/mL (insoluble)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.5038 mL 12.5188 mL 25.0376 mL
5 mM 0.5008 mL 2.5038 mL 5.0075 mL
10 mM 0.2504 mL 1.2519 mL 2.5038 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: 2.5 mg/mL (6.26 mM); Suspended solution; Need ultrasonic

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: 2.5 mg/mL (6.26 mM); Suspended solution; Need ultrasonic

  • 3.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.5 mg/mL (6.26 mM); Clear solution

*All of the co-solvents are provided by MCE.
References
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  • Molarity Calculator

  • Dilution Calculator

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This equation is commonly abbreviated as: C1V1 = C2V2

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Keywords:

MRS-3777 hemioxalateAdenosine ReceptorP1 receptorInhibitorinhibitorinhibit

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Product Name:
MRS-3777 hemioxalate
Cat. No.:
HY-110037
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