NEU-1017
NEU-1017 is a broad-spectrum antiparasitic agent. NEU-1017 inhibits T. brucei, L. major, and P. falciparum with EC50 values of 210 nM, 240 nM, and 3 nM, respectively. X
For research use only. We do not sell to patients.
- CAS No.: 1800426-38-3
- Formula: C33H31ClFN5O3S
- Molecular Weight:632.15
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Parasite Isoforms
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Biological Activity
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| RAW264.7 | EC50 |
0.24 μM
Compound: 68, NEU-1017
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Antiparasite activity against luciferase-expressing Leishmania major amastigotes isolated from infected in mouse RAW264.7 cells assessed as growth inhibition incubated for 96 hrs by luciferase reporter gene assay
Antiparasite activity against luciferase-expressing Leishmania major amastigotes isolated from infected in mouse RAW264.7 cells assessed as growth inhibition incubated for 96 hrs by luciferase reporter gene assay
|
[PMID: 26087257] |
Chemical Information
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CAS No. 1800426-38-3
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Molecular Weight 632.15
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Formula C33H31ClFN5O3S
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SMILES
CN1CCCN(S(=O)(C2=CC=C(C3=CC(N=NC=C4NC5=CC(Cl)=C(OCC6=CC(F)=CC=C6)C=C5)=C4C=C3)C=C2)=O)CC1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)