1. Metabolic Enzyme/Protease
  2. Drug Metabolite
  3. O-Desmethyl apixaban

O-Desmethyl apixaban 

Cat. No.: HY-100655
Handling Instructions

O-Desmethyl apixaban is a metabolite of Apixaban (BMS-562247-01). Apixaban is a highly selective, reversible inhibitor of Factor Xa with Ki of 0.08 nM and 0.17 nM in human and rabbit, respectively.

For research use only. We do not sell to patients.

O-Desmethyl apixaban Chemical Structure

O-Desmethyl apixaban Chemical Structure

CAS No. : 503612-76-8

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Description

O-Desmethyl apixaban is a metabolite of Apixaban (BMS-562247-01)[1]. Apixaban is a highly selective, reversible inhibitor of Factor Xa with Ki of 0.08 nM and 0.17 nM in human and rabbit, respectively[2].

Molecular Weight

445.47

Formula

C₂₄H₂₃N₅O₄

CAS No.

503612-76-8

SMILES

O=C(C1=NN(C2=CC=C(O)C=C2)C3=C1CCN(C4=CC=C(N5C(CCCC5)=O)C=C4)C3=O)N

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

O-Desmethyl apixabanDrug MetabolitemetabolitethromboembolicdiseasesInhibitorinhibitorinhibit

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O-Desmethyl apixaban
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