1. GPCR/G Protein Neuronal Signaling
  2. mAChR
  3. Parapenzolate bromide

Parapenzolate bromide, an antispasmodic, is an orally active mAChR antagonist. Parapenzolate bromide is an anticholinergic agent.

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Parapenzolate bromide Chemical Structure

Parapenzolate bromide Chemical Structure

CAS No. : 5634-41-3

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Description

Parapenzolate bromide, an antispasmodic, is an orally active mAChR antagonist. Parapenzolate bromide is an anticholinergic agent[1][2].

In Vivo

Parapenzolate bromide (10 mg/kg, p.o. or i.v.) shows a significant analgesic effect in mice[1].
Parapenzolate bromide (0.5 mg/kg, i.v.) exhibits a spasmolytic activity in isolated gall bladder from guinea pigs[2].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Mice[1]
Dosage: 10 mg/kg
Administration: Oral administration (p.o.) or intravenous injection (i.v.)
Result: Prolonged the time until death in convulsive mice.
Animal Model: Guinea pigs[2]
Dosage: 0.5 mg/kg
Administration: Intravenous injection (i.v.)
Result: Antagonized contractions induced by acetylcholine (100 μg/kg, i.v.)
Molecular Weight

420.34

Formula

C21H26BrNO3

CAS No.
SMILES

C[N+](CC1)(C)CCC1OC(C(C2=CC=CC=C2)(C3=CC=CC=C3)O)=O.[Br-]

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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Parapenzolate bromide Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Parapenzolate bromide
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HY-105771
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