PPARγ/δ modulator 1
PPARγ/δ modulator 1 (compound 3e) is a potent PPAR modulator. PPARγ/δ modulator 1 is a PPARδ antagonist and a PPARγ partial agonist , with Ki values of 14.4 nM and 5.31 μM, respectively. PPARγ/δ modulator 1 has the EC50 of 7.3 and 12.6 μM for PPARδ corepression and adiponectin production, respectively.
For research use only. We do not sell to patients.
- CAS No.: 2089159-00-0
- Formula: C18H18ClIN6O3Se
- Molecular Weight:607.69
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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PPARδ 14.4 nM (Ki) |
PPARγ 5.31 μM (Ki) |
Chemical Information
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CAS No. 2089159-00-0
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Molecular Weight 607.69
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Formula C18H18ClIN6O3Se
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SMILES
O[C@H]1[C@H]([C@@H]([Se][C@@H]1C(NC)=O)N2C3=C(N=C2)C(NCC4=CC=CC(I)=C4)=NC(Cl)=N3)O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
PPARγ/δ modulator 1 Related Classifications
HY-147757 Related Classifications
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