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    PROTAC
  2. Estrogen Receptor/ERR
    PROTAC
  3. PROTAC ER Degrader-2

PROTAC ER Degrader-2 

Cat. No.: HY-128528
Handling Instructions

PROTAC ER Degrader-2 is an intermediate for synthesis of PAC. PAC, consists the ADCs linker and PROTACs, conjugated to an antibody. PAC extracts from patent WO2017201449A1, compound LP2. PAC conjugated to an antibody is a more marked estrogen receptor-alpha (ERα) degrader compared to PROTAC (without Ab).

For research use only. We do not sell to patients.

PROTAC ER Degrader-2 Chemical Structure

PROTAC ER Degrader-2 Chemical Structure

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10 mg USD 850 Get quote

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Description

PROTAC ER Degrader-2 is an intermediate for synthesis of PAC. PAC, consists the ADCs linker and PROTACs, conjugated to an antibody. PAC extracts from patent WO2017201449A1, compound LP2. PAC conjugated to an antibody is a more marked estrogen receptor-alpha (ERα) degrader compared to PROTAC (without Ab)[1].

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
Molecular Weight

1581.85

Formula

C₈₉H₁₀₄N₁₂O₁₅

SMILES

CC/C(C1=CC=CC=C1)=C(C2=CC=C(OCCN(C)C(COCCOCCNC(C3=CC=C(C(N4[[email protected]@H](C)[[email protected]](NC([[email protected]](C)N(C(OC(C)(C)C)=O)C)=O)C(N(CC5=C(OC)C=CC6=C5C=CC=C6)C7=C4C=C(C#N)C=C7)=O)=O)C=C3)=O)=O)C=C2)\C8=CC=C(OCC9=CC=C(NC([[email protected]@H](NC([[email protected]](C(C)C)N)=O)CCCNC(N)=O)=O)C=C9)C=C8

Shipping

Room temperature in continental US; may vary elsewhere

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This equation is commonly abbreviated as: C1V1 = C2V2

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C1   V1   C2   V2

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Product Name:
PROTAC ER Degrader-2
Cat. No.:
HY-128528
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PROTAC ER Degrader-2

Cat. No.: HY-128528