PSB-KK1415
Based on 1 Customer Validation
PSB-KK1415 is a selective agonist for human orphan G protein-coupled receptor GPR18, with EC50 of 19.1 nM.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度: 99.92%
- CAS 番号: 885896-26-4
- 分子式: C24H23ClN6O2
- 分子量:462.93
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保管条件:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
生物活性
IC50: 19.1 nM (GPR18)
化学情報
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CAS 番号 885896-26-4
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性状 Solid
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分子量 462.93
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分子式 C24H23ClN6O2
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Color White to off-white
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SMILES
CN1C2=C(C(N(C1=O)C)=O)N(C(NCCC3=CNC4=C3C=CC=C4)=N2)CC5=CC=C(C=C5)Cl
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
溶剤 & 溶解度
DMSO : 100 mg/mL (216.02 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
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データシート (275 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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取扱説明書 (2659 KB)
参考文献
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.1602 mL | 10.8008 mL | 21.6015 mL | 54.0038 mL |
| 5 mM | 0.4320 mL | 2.1602 mL | 4.3203 mL | 10.8008 mL | |
| 10 mM | 0.2160 mL | 1.0801 mL | 2.1602 mL | 5.4004 mL | |
| 15 mM | 0.1440 mL | 0.7201 mL | 1.4401 mL | 3.6003 mL | |
| 20 mM | 0.1080 mL | 0.5400 mL | 1.0801 mL | 2.7002 mL | |
| 25 mM | 0.0864 mL | 0.4320 mL | 0.8641 mL | 2.1602 mL | |
| 30 mM | 0.0720 mL | 0.3600 mL | 0.7201 mL | 1.8001 mL | |
| 40 mM | 0.0540 mL | 0.2700 mL | 0.5400 mL | 1.3501 mL | |
| 50 mM | 0.0432 mL | 0.2160 mL | 0.4320 mL | 1.0801 mL | |
| 60 mM | 0.0360 mL | 0.1800 mL | 0.3600 mL | 0.9001 mL | |
| 80 mM | 0.0270 mL | 0.1350 mL | 0.2700 mL | 0.6750 mL | |
| 100 mM | 0.0216 mL | 0.1080 mL | 0.2160 mL | 0.5400 mL |