2. GPCR/G Protein Neuronal Signaling
  3. Opioid Receptor
  4. SCH 221510

SCH 221510 is a potent, orally active and selective NOP (nociceptin opioid receptor) agonist, with an EC50 of 12 nM and Ki of 0.3 nM. SCH 221510 shows an anxiolytic-like effect.

For research use only. We do not sell to patients.

SCH 221510 Chemical Structure

SCH 221510 Chemical Structure

CAS No. : 322473-89-2

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SCH 221510 Related Antibodies

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Description

SCH 221510 is a potent, orally active and selective NOP (nociceptin opioid receptor) agonist, with an EC50 of 12 nM and Ki of 0.3 nM. SCH 221510 shows an anxiolytic-like effect[1].

IC50 & Target

EC50: 12 nM (NOP)[1]
Molecular Weight

397.55

Formula

C28H31NO
CAS No.
SMILES

O[C@](C[C@H]1CC2)(C3=CC=CC=C3)C[C@H]2N1C(C4=C(C=CC=C4)C)C5=C(C=CC=C5)C
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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SCH 221510 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

SCH 221510322473-89-2SCH221510SCH-221510Opioid Receptororally activehigh affinityanxiolytic-like activityOpioid receptorInhibitorinhibitorinhibit

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SCH 221510
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HY-107722
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