14 Results for "

PKA catalytic subunit

" in MedChemExpress (MCE) Product Catalog:
Products (14)

14 Results for "PKA catalytic subunit" in MCE Product Catalog:

5
5 Cited Publications
Art. -Nr.: HY-P1290
CAS. Nr.: 121932-06-7
Synonyms: PKI-(6-22)-amide
Target:  

PKA

Forschungsgebiete:  

Neurological Disease

PKA Inhibitor Fragment (6-22) amide is a highly potent and specific competitive inhibitor of PKA, with Ki values of 1.7 nM and 1.6 nM against human and bovine PKA catalytic subunits, respectively. The IC50 of PKA Inhibitor Fragment (6-22) amide targeting bovine PKA is 8.6 nM. PKA Inhibitor Fragment (6-22) amide effectively abolishes PKA activity in mouse brain and spinal cord, and exerts in vivo efficacy via intracerebroventricular administration. PKA Inhibitor Fragment (6-22) amide significantly reverses low-dose morphine analgesic tolerance in mice and blocks photoaffinity labeling of cAMP-dependent protein kinase. PKA Inhibitor Fragment (6-22) amide can be applied to research in fields related to the mechanism of morphine analgesic tolerance and skin wound healing .
loading...
    loading...
1
1 Cited Publications
Art. -Nr.: HY-115732
CAS. Nr.: 179985-52-5
Reinheit:  99.82%
Target:  

PKA

Forschungsgebiete:  

Inflammation/Immunology

PKA-IN-1 is a potent and selective cyclic AMP-dependent protein kinase (PKA) catalytic subunit (cAK) inhibitor with an IC50 of 0.03 μM. PKA-IN-1 inhibits cAK in a fashion that is competitive with respect to ATP as substrate .
loading...
    loading...
Art. -Nr.: HY-P2629
CAS. Nr.: 128022-93-5
Target:  

PKA

Forschungsgebiete:  

Infection

PKI (5-22) is a specific inhibitory peptide targeting the catalytic subunit of protein kinase A (PKA) and contains the active region of PKI. PKI (5-22) inhibits the enzymatic activity of the PKA catalytic subunit-like protein in Trypanosoma equiperdum. PKI (5-22) can be used in the research of trypanosomiasis .
loading...
    loading...
Art. -Nr.: HY-P81127
Synonyms: PRKACA/PRKACB; PRKACA + PRKACB; PKA alpha + beta; PKA alpha; PKA beta; cAMP dependent protein kinase alpha catalytic subunit; cAMP dependent protein kinase beta catalytic subunit; cAMP dependent protein kinase catalytic subunit alpha; cAMP dependent protein kinase catalytic subunit beta; DKFZp781I2452; MGC102831; MGC41879; MGC48865; MGC9320; PKA C alpha; PKA C beta; PKACA; PKACB; PRKACA; PRKACB; Protein kinase A catalytic subunit alpha; Protein kinase A catalytic subunit; Protein kinase A catalytic subunit beta; Protein kinase cAMP dependent catalytic alpha; Protein kinase cAMP dependent catalytic beta; cAMP dependent protein kinase catalytic subunit alpha isoform 1; cAMP-dependent protein kinase catalytic subunit alpha; KAPCA_HUMAN; KAPCB_HUMAN; PKA C alpha; PKA C-alpha; PKACA; PRKACA; Protein kinase A catalytic subunit; Protein kinase cAMP dependent catalytic alpha.

Host:  

Rabbit

Application:  

WB, ICC/IF

Reactivity:  

Human, Mouse, Rat

loading...
    loading...
Art. -Nr.: HY-P810621
Synonyms: PRKACA/PRKACB; PRKACA + PRKACB; PKA alpha + beta; PKA alpha; PKA beta; cAMP dependent protein kinase alpha catalytic subunit; cAMP dependent protein kinase beta catalytic subunit; cAMP dependent protein kinase catalytic subunit alpha; cAMP dependent protein kinase catalytic subunit beta; DKFZp781I2452; MGC102831; MGC41879; MGC48865; MGC9320; PKA C alpha; PKA C beta; PKACA; PKACB; PRKACA; PRKACB; Protein kinase A catalytic subunit alpha; Protein kinase A catalytic subunit; Protein kinase A catalytic subunit beta; Protein kinase cAMP dependent catalytic alpha; Protein kinase cAMP dependent catalytic beta; cAMP dependent protein kinase catalytic subunit alpha isoform 1; cAMP-dependent protein kinase catalytic subunit alpha; KAPCA_HUMAN; KAPCB_HUMAN; PKA C alpha; PKA C-alpha; PKACA; PRKACA; Protein kinase A catalytic subunit; Protein kinase cAMP dependent catalytic alpha.

Host:  

Rabbit

Application:  

WB

Reactivity:  

Human, Mouse, Rat

loading...
    loading...
Art. -Nr.: HY-P810911
Synonyms: cAMP-dependent protein kinase catalytic subunit beta, PKA C-beta, PRKACB

Host:  

Rabbit

Application:  

WB, IHC-P

Reactivity:  

Human, Mouse, Rat

loading...
    loading...
Art. -Nr.: HY-P81981
Synonyms: PRKACG; cAMP-dependent protein kinase catalytic subunit gamma; PKA C-gamma

Host:  

Rabbit

Application:  

WB

Reactivity:  

Human, Mouse, Rat

loading...
    loading...
Art. -Nr.: HY-P86462
Synonyms: PRKACA; PKACA; cAMP-dependent protein kinase catalytic subunit alpha; PKA C-alpha

Host:  

Rabbit

Application:  

WB, IHC-P, ICC/IF, IP, ELISA

Reactivity:  

Human, Mouse, Rat

loading...
    loading...
Art. -Nr.: HY-P701753
Reinheit:  ≥ 90%, as determined by reducing SDS-PAGE.
Synonyms: PRKACA; cAMP-dependent protein kinase catalytic subunit alpha; PKA C-alpha
Species:  
Source:  
loading...
    loading...
Art. -Nr.: HY-P81981A
Synonyms: PRKACG; cAMP-dependent protein kinase catalytic subunit gamma; PKA C-gamma

Host:  

Rabbit

Application:  

WB

Reactivity:  

Human, Mouse, Rat

loading...
    loading...
Art. -Nr.: HY-P87988
Synonyms: cAMP-dependent protein kinase catalytic subunit gamma, PKA C-gamma, PRKACG

Host:  

Rabbit

Application:  

WB, IHC-P, IHC-F, IF-Tissue

Reactivity:  

Human, Mouse, Rat

loading...
    loading...
Art. -Nr.: HY-P702637
Reinheit:  ≥ 80%, as determined by reducing SDS-PAGE.
Synonyms: PRKACB; protein kinase, cAMP-dependent, catalytic, beta; cAMP-dependent protein kinase catalytic subunit beta; PKACb; PKA C-beta; protein kinase A catalytic subunit beta; cAMP-dependent protein kinase catalytic beta subunit isoform 4ab; PKACB; MGC9320; MGC41879; DKFZp781I2452
Species:  
Source:  
loading...
    loading...
Art. -Nr.: HY-P702638
Reinheit:  ≥ 80%, as determined by reducing SDS-PAGE.
Synonyms: PRKACG; protein kinase, cAMP-dependent, catalytic, gamma; cAMP-dependent protein kinase catalytic subunit gamma; PKACg; PKA C-gamma; serine(threonine) protein kinase; KAPG
Species:  
Source:  
loading...
    loading...
Art. -Nr.: HY-P705862
Reinheit:  ≥ 90%, as determined by reducing SDS-PAGE.
Synonyms: PRKACA; cAMP-dependent protein kinase catalytic subunit alpha; PKA C-alpha
Species:  
Source:  
loading...
    loading...
  • 1