1. Membrane Transporter/Ion Channel
    Neuronal Signaling
  2. GABA Receptor
  3. TP003

TP003 

Cat. No.: HY-103512
Handling Instructions

TP003 is a non-selective benzodiazepine site agonist with EC50s of 20.3, 10.6, 3.24, 5.64 nM for α1β2γ2, α2β3γ2, α3β3γ2, α5β2γ2, respectively. TP003 induces anxiolysis via α2GABAA receptors.

For research use only. We do not sell to patients.

TP003 Chemical Structure

TP003 Chemical Structure

CAS No. : 628690-75-5

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Description

TP003 is a non-selective benzodiazepine site agonist with EC50s of 20.3, 10.6, 3.24, 5.64 nM for α1β2γ2, α2β3γ2, α3β3γ2, α5β2γ2, respectively. TP003 induces anxiolysis via α2GABAA receptors[1].

Molecular Weight

407.39

Formula

C23H16F3N3O

CAS No.
SMILES

N#CC1=CC(F)=CC=C1C2=CC(C3=CN=C4C(F)=C(C(C)(O)C)C=CN43)=CC=C2F

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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TP003
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