UniPR1454
UniPR1454 targets EphA2 receptor, inhibits the EphA2-ephrin A1 interaction with an IC50 of 2.6 μM. UniPR1454 inhibits the proliferation of glioblastoma cell U251.
For research use only. We do not sell to patients.
- Formula: C43H53F3N2O6S
- Molecular Weight:782.95
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
|
EphA4 4.2 μM (IC50) |
EphA5 9.3 μM (IC50) |
EphA6 10 μM (EC50) |
EphA1 11 μM (IC50) |
EphA8 13 μM (IC50) |
EphA7 15 μM (IC50) |
Chemical Information
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Molecular Weight 782.95
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Formula C43H53F3N2O6S
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SMILES
C[C@]12[C@]([H])([C@]3([C@@]([H])([C@]4(C)C(C[C@@H](O)CC4)=CC3)CC2)[H])CC[C@@]1([C@@H](CCC(N[C@H](CC(O)=O)CC5=CN(C6=C5C=CC=C6)S(=O)(C7=CC=C(C=C7)C(F)(F)F)=O)=O)C)[H]
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)