UVI3502
UVI3502 is a cannabinoid receptor 1 (CB1) antagonist with an IC50 value of 4641 nM for CB1 and approximately 16200 nM for CB2. UVI3502 blocks Gi/o protein coupling induced by the agonist CP55,940. UVI3502 is promising for research of endocannabinoid system-related diseases in the central nervous system (such as cognitive impairment and neurodegenerative diseases).
For research use only. We do not sell to patients.
- Formula: C25H24N2O6
- Molecular Weight:448.47
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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CB1 4641 nM (IC50) |
CB2 16200 nM (IC50) |
Chemical Information
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Molecular Weight 448.47
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Formula C25H24N2O6
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SMILES
COC1=CC2=C(N(C(OCC)=O)C(C(C=C(C)C=C3)=C3NC/4=O)=C2C4=C\C(OCC)=O)C=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)