5-HT4 antagonist 1
Based on 1 Customer Validation
5-HT4 antagonist 1 is a 5-HT4 receptor antagonist with a pKi of 9.6.
For research use only. We do not sell to patients.
- Purity: 98.95%
- CAS No.: 261766-73-8
- Formula: C23H36N4O5S
- Molecular Weight:480.62
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Storage:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
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Biological Activity
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Chemical Information
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Solvent & Solubility
- Purity & Documentation
- References
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Help & FAQs
All 5-HT Receptor Isoforms
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Biological Activity
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5-HT4 Receptor 9.6 (pKi) |
5-HT4 antagonist 1 (compound 6b) is a 5-HT4 receptor antagonist with a pKi of 9.6.
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 261766-73-8
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Appearance Solid
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Molecular Weight 480.62
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Formula C23H36N4O5S
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Color Light brown to brown
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SMILES
O=C(C1=C2OCCOC2=CC=C1)NCC3CCN(CCCS(=O)(N4CCN(C)CC4)=O)CC3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
DMSO : 20 mg/mL (41.61 mM; ultrasonic and warming and adjust pH to 3 with HCl and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (270 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
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| DMSO | 1 mM | 2.0806 mL | 10.4032 mL | 20.8065 mL | 52.0161 mL |
| 5 mM | 0.4161 mL | 2.0806 mL | 4.1613 mL | 10.4032 mL | |
| 10 mM | 0.2081 mL | 1.0403 mL | 2.0806 mL | 5.2016 mL | |
| 15 mM | 0.1387 mL | 0.6935 mL | 1.3871 mL | 3.4677 mL | |
| 20 mM | 0.1040 mL | 0.5202 mL | 1.0403 mL | 2.6008 mL | |
| 25 mM | 0.0832 mL | 0.4161 mL | 0.8323 mL | 2.0806 mL | |
| 30 mM | 0.0694 mL | 0.3468 mL | 0.6935 mL | 1.7339 mL | |
| 40 mM | 0.0520 mL | 0.2601 mL | 0.5202 mL | 1.3004 mL |
5-HT4 antagonist 1 Related Classifications
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