5-HT2C antagonist 1
5-HT2C antagonist 1 (Compound 45) is a selective and orally active 5-HT2C receptor antagonist with a pKi of 8.0. 5-HT2C antagonist 1 can effectively antagonize the erection of the rat penis induced by mCPP. 5-HT2C antagonist 1 can be used for the researches of neurological disease and endocrinology, such as anxiety.
For research use only. We do not sell to patients.
- CAS No.: 204650-40-8
- Formula: C17H23NO3
- Molecular Weight:289.37
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All 5-HT Receptor Isoforms
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Biological Activity
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5-HT2C Receptor 8.0 (pKi) |
Chemical Information
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CAS No. 204650-40-8
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Molecular Weight 289.37
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Formula C17H23NO3
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SMILES
OC1=C2C([C@@]3([H])[C@](CCN(C3)C)([H])CC2=O)=CC(OC)=C1CC
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)