5-HT4R agonist-2
5-HT4R agonist-2 (Compound 4) is a selective 5-HT4R agonist with an EC50 value of 0.41 nM. 5-HT4R agonist-2 can significantly enhance whole gut and colonic transit, increase fecal output and water content, while maintaining minimal systemic absorption, and it shows promise for the research of chronic idiopathic constipation.
For research use only. We do not sell to patients.
- Formula: C60H96Cl2N12O12
- Molecular Weight:1248.38
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All 5-HT Receptor Isoforms
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Biological Activity
Chemical Information
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Molecular Weight 1248.38
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Formula C60H96Cl2N12O12
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SMILES
O=C(CCCCCN1CCC(CNC(C2=C(OCC3)C3=C(N)C(Cl)=C2)=O)CC1)NCCOCCOCCNC(NCCCCNC(NCCOCCOCCNC(CCCCCN4CCC(CNC(C5=C(OCC6)C6=C(N)C(Cl)=C5)=O)CC4)=O)=O)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)