1. GPCR/G Protein
    Neuronal Signaling
  2. Melatonin Receptor
    5-HT Receptor
  3. 7-Desmethyl-3-hydroxyagomelatine

7-Desmethyl-3-hydroxyagomelatine (Synonyms: 3-Hydroxy-7-desmethyl agomelatine)

Cat. No.: HY-133112
Handling Instructions

7-Desmethyl-3-hydroxyagomelatine (3-Hydroxy-7-desmethyl agomelatine), a metabolite of Agomelatine, has less activity than Agomelatine. Agomelatine is a melatonergic (MT1 and MT2) agonist and serotonergic (5HT2C) antagonist.

For research use only. We do not sell to patients.

7-Desmethyl-3-hydroxyagomelatine Chemical Structure

7-Desmethyl-3-hydroxyagomelatine Chemical Structure

CAS No. : 166527-00-0

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Description

7-Desmethyl-3-hydroxyagomelatine (3-Hydroxy-7-desmethyl agomelatine), a metabolite of Agomelatine, has less activity than Agomelatine[1]. Agomelatine is a melatonergic (MT1 and MT2) agonist and serotonergic (5HT2C) antagonist[1][2].

IC50 & Target[1][2]

MT1

 

MT2

 

5-HT2C Receptor

 

Molecular Weight

245.27

Formula

C₁₄H₁₅NO₃

CAS No.

166527-00-0

SMILES

CC(NCCC1=C2C=C(O)C=CC2=CC(O)=C1)=O

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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

7-Desmethyl-3-hydroxyagomelatine3-Hydroxy-7-desmethyl agomelatineMelatonin Receptor5-HT ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorMT1MT2Agonist5-HT2CAntagonistdepressivedisorderInhibitorinhibitorinhibit

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7-Desmethyl-3-hydroxyagomelatine
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HY-133112
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