2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. iGluR
  4. AMPA receptor modulator-1

AMPA receptor modulator-1 is a potent, orally active and selective AMPAR regulatory protein TARP γ-8 negative modulator with a pIC50 of 9.7, more selective over GluA1/γ-2 (pIC50=5).

For research use only. We do not sell to patients.

AMPA receptor modulator-1 Chemical Structure

AMPA receptor modulator-1 Chemical Structure

CAS No. : 2036074-41-4

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AMPA receptor modulator-1 Related Antibodies

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Description

AMPA receptor modulator-1 is a potent, orally active and selective AMPAR regulatory protein TARP γ-8 negative modulator with a pIC50 of 9.7, more selective over GluA1/γ-2 (pIC50=5)[1].

IC50 & Target

pIC50: 9.7 (TARP γ-8)[1]
Molecular Weight

341.71

Formula

C16H11ClF3NO2
CAS No.
SMILES

ClC1=C(C2=CC(C)=C(NC(C3)=O)C3=C2)C(OC(F)(F)F)=CC=C1
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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AMPA receptor modulator-1 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

AMPA receptor modulator-12036074-41-4AMPA receptor modulator1AMPA receptor modulator 1iGluRIonotropic glutamate receptorsInhibitorinhibitorinhibit

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AMPA receptor modulator-1
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HY-112699
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