1. Membrane Transporter/Ion Channel
    Neuronal Signaling
  2. iGluR
  3. AMPA receptor modulator-1

AMPA receptor modulator-1 

Cat. No.: HY-112699
Handling Instructions

AMPA receptor modulator-1 is a potent, orally active and selective AMPAR regulatory protein TARP γ-8 negative modulator with a pIC50 of 9.7, more selective over GluA1/γ-2 (pIC50=5).

For research use only. We do not sell to patients.

AMPA receptor modulator-1 Chemical Structure

AMPA receptor modulator-1 Chemical Structure

CAS No. : 2036074-41-4

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Description

AMPA receptor modulator-1 is a potent, orally active and selective AMPAR regulatory protein TARP γ-8 negative modulator with a pIC50 of 9.7, more selective over GluA1/γ-2 (pIC50=5)[1].

IC50 & Target

pIC50: 9.7 (TARP γ-8)[1]

Molecular Weight

341.71

Formula

C₁₆H₁₁ClF₃NO₂

CAS No.

2036074-41-4

SMILES

ClC1=C(C2=CC(C)=C(NC(C3)=O)C3=C2)C(OC(F)(F)F)=CC=C1

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

AMPA receptor modulator-1AMPA receptor modulator1AMPA receptor modulator 1iGluRIonotropic glutamate receptorsInhibitorinhibitorinhibit

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AMPA receptor modulator-1
Cat. No.:
HY-112699
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