1. GPCR/G Protein
  2. GPR40

GPR40 agonist 1 

Cat. No.: HY-111359
Handling Instructions

GPR40 agonist 1 is a potent and novel GPR40 full agonist with an EC50 of 2 nM and 17 nM for hGPR40 and rGPR40, respectively.

For research use only. We do not sell to patients.

GPR40 agonist 1 Chemical Structure

GPR40 agonist 1 Chemical Structure

CAS No. : 1853982-41-8

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  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

GPR40 agonist 1 is a potent and novel GPR40 full agonist with an EC50 of 2 nM and 17 nM for hGPR40 and rGPR40, respectively.

IC50 & Target

EC50: 2 nM (hGPR40), 17 nM (rGPR40)[1]

Solvent & Solubility
In Vitro: 

10 mM in DMSO

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.0853 mL 10.4267 mL 20.8533 mL
5 mM 0.4171 mL 2.0853 mL 4.1707 mL
10 mM 0.2085 mL 1.0427 mL 2.0853 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

479.54

Formula

C₂₇H₃₀FN₃O₄

CAS No.

1853982-41-8

SMILES

COC1=NC=C(F)C(C2=C(CC(C)C)N=C(COC3=CC=CC([[email protected]](C4CC4)CC(O)=O)=C3)C=N2)=C1

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
GPR40 agonist 1
Cat. No.:
HY-111359
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GPR40 agonist 1

Cat. No.: HY-111359