1. Metabolic Enzyme/Protease
  2. Fatty Acid Synthase (FAS)

FASN inhibitor 1 

Cat. No.: HY-U00436
Handling Instructions

FASN inhibitor 1 is a fatty acid synthase (FASN) inhibitor extracted from patent US20170119786A1, compound 242A.

For research use only. We do not sell to patients.

FASN inhibitor 1 Chemical Structure

FASN inhibitor 1 Chemical Structure

CAS No. : 2097262-60-5

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  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

FASN inhibitor 1 is a fatty acid synthase (FASN) inhibitor extracted from patent US20170119786A1, compound 242A.

IC50 & Target

FASN[1]

In Vitro

Human PBMC and monocytes in cell cultures are stimulated with lipopolysaccharide (LPS), a Toll 4 receptor agonist, or lipoteichoic acid (LTA), a Toll 2 receptor agonist. Stimulation with either LPS or LTA plus DMSO, the solvent for FASN inhibitor 1 (Compound 242A), results in secretion of IL-1 beta. FASN inhibitor 1 treatment of PBMC, which is a mixed population of mononuclear cells including both lymphocytes and monocytes, reduces the level of IL-1 beta resulting from either LPS or LTA stimulation. For monocytes, FASN inhibitor 1 treatment reduces the level of IL-1 beta resulting from LTA stimulation whereas there is only a slight reduction after LPS stimulation[1].

References
Molecular Weight

384.47

Formula

C₂₄H₂₄N₄O

CAS No.

2097262-60-5

SMILES

N#CC1=CC=C(C2CN(C(C3=CC(C4=C(C)C(C)=NN4)=C(C)C=C3C)=O)C2)C=C1

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

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× = ×
C1   V1   C2   V2

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Product Name:
FASN inhibitor 1
Cat. No.:
HY-U00436
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FASN inhibitor 1

Cat. No.: HY-U00436