1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. DYRK
  4. DYRK Degrader

DYRK Degrader

DYRK Degraders (2):

Cat. No. Product Name Effect Purity
  • HY-161597
    PROTAC DYRK2 degrader 1
    Degrader
    PROTAC DYRK2 degrader 1 is a DYRK2 PROTAC degrader with DC50 values of 1.607 μM (MDA-MB-231 cells) and 3.265 μM (HeLa cells), respectively. PROTAC DYRK2 degrader 1 induces DYRK2 degradation via the ubiquitin-proteasome system. It is applicable to the research of triple-negative breast cancer and cervical cancer.
  • HY-161598
    DYRK2 ligand 1
    Degrader
    DYRK2 ligand 1 is a target protein ligand of PROTAC DYRK2 degrader 1 (HY-161597). DYRK2 ligand 1 can be used to study cancer.