iGluR
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iGluR Related Products (456)
Related Products (456)
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(Rac)-Lanicemine (Standard)
0 ImagesCat. No.: HY-108235BRCAS No.: 61890-25-3Synonyms: (Rac)-AZD6765 (Standard)(Rac)-Lanicemine (Standard) is the analytical standard of (Rac)-Lanicemine. This product is intended for research and analytical applications. (Rac)-Lanicemine ((Rac)-AZD6765) is the racemate of Lanicemine. Lanicemine (AZD6765) is a low-trapping NMDA channel blocker (Ki of 0.56-2.1 μM for NMDA receptor; IC50s of 4-7 μM and 6.4 μM in CHO and Xenopus oocyte cells, respectively). Antidepressant effects.
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Gacyclidine hydrochloride
0 ImagesCat. No.: HY-15410ACAS No.: 131774-33-9Gacyclidine hydrochloride, a non competitive N-methyl-D-aspartate (NMDA) antagonist, can be used in the study of spinal cord injuries.
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ZL006 (Standard)
0 ImagesCat. No.: HY-100456RCAS No.: 1181226-02-7
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Omberacetam (Standard)
0 ImagesSynonyms: GVS-111 (Standard); SGS-111 (Standard)Omberacetam (Standard) is the analytical standard of Omberacetam. This product is intended for research and analytical applications. Omberacetam (GVS-111) is a medication promoted and prescribed in Russia and neighbouring countries as a nootropic.
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Kynurenic acid sodium (Standard)
0 ImagesKynurenic acid (sodium) (Standard) is the analytical standard of Kynurenic acid (sodium). This product is intended for research and analytical applications. Kynurenic acid sodium, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid sodium is also an agonist of GPR35/CXCR8.
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Piracetam-d8
0 ImagesCat. No.: HY-B0585SCAS No.: 1329799-64-5Piracetam-d8 (UCB-6215-d8) is the deuterium labeled Piracetam. Piracetam (UCB-6215) is a cyclic derivative of the neurotransmitter gamma-aminobutyric acid (GABA), used in treatment of a wide range of cognitive disorders.
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Mephenesin (Standard)
0 ImagesMephenesin (Standard) is the analytical standard of Mephenesin. This product is intended for research and analytical applications. Mephenesin is an NMDA receptor antagonist and Mephenesin is a central muscle relaxant.
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Apimostinel (Standard)
0 ImagesCat. No.: HY-102053RCAS No.: 1421866-48-9Synonyms: NRX-1074 (Standard); AGN-241660 (Standard)Apimostinel (Standard) is the analytical standard of Apimostinel (HY-102053). This product is intended for research and analytical applications. Apimostinel (NRX-1074; AGN-241660) is an orally active NMDA receptor partial agonist.
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Topiramate-13C6-1
0 ImagesCat. No.: HY-B0122SS1Synonyms: McN 4853-13C6-1; RWJ 17021-13C6-1
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7-Chlorokynurenic acid (Standard)
0 ImagesSynonyms: 7-CKA (Standard)7-Chlorokynurenic acid (Standard) is the analytical standard of 7-Chlorokynurenic acid. This product is intended for research and analytical applications. 7-Chlorokynurenic acid (7-CKA) is a potent and selective antagonist of the glycine B coagonist site of the N-methyl-D-aspartate (NMDA) receptor (IC50=0.56 μM). 7-Chlorokynurenic acid is also a potent inhibitor of the reuptake of glutamate into synaptic vesicles with a Ki of 0.59 μM. 7-Chlorokynurenic acid has potent antinociceptive actions after neuraxial delivery.
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DL-AP5 (Standard)
0 ImagesCat. No.: HY-100714RCAS No.: 76326-31-3Synonyms: 2-APV (Standard); DL-2-Amino-5-phosphonovaleric acid (Standard)DL-AP5 (Standard) is the analytical standard of DL-AP5. This product is intended for research and analytical applications. DL-AP5 (2-APV) is a competitive NMDA (N-methyl-D-aspartate) receptor antagonist. DL-AP5 shows significantly antinociceptive activity. DL-AP5 specifically blocks on channels in the rabbit retina.
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Flupirtine Maleate (Standard)
0 ImagesSynonyms: D 9998 Maleate (Standard)Flupirtine Maleate (Standard) is the analytical standard of Flupirtine Maleate (HY-17001). This product is intended for research and analytical applications. Flupirtine Maleate is an orally active, blood-brain barrier-crossing non-opioid analgesic and neuroprotective agent. Flupirtine Maleate is a neuronal potassium channel opener (Kv7 activator), a NMDA receptor antagonist and a GABA receptor activator. Flupirtine Maleate stabilizes blood-brain-barrier integrity, reduces oxidative stress and brain leukocyte infiltration, enhances angioneurogenesis, suppresses calcium influx, stabilizes neuronal resting membrane potential, and counteracts focal cerebral ischemia. Flupirtine Maleate exhibits analgesic, muscle relaxant properties, protects neurons from excitotoxic, ischemic, or cytokine-mediated death. Flupirtine Maleate functions as a non-opioid analgesic without antipyretic or antiphlogistic properties, shows no relevant affinity to opiate receptor. Flupirtine Maleate can be used for the research of focal cerebral ischemia, pain, Alzheimer’s disease, or multiple sclerosis.
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GRIN2A modulator-1
0 ImagesCat. No.: HY-180866CAS No.: 898203-28-6GRIN2A modulator-1 is a GRIN2A modulator.
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Sepimostat (Standard)
0 ImagesCat. No.: HY-136299RCAS No.: 103926-64-3Synonyms: FUT-187 free base (Standard)Sepimostat (Standard) is the analytical standard of Sepimostat. This product is intended for research and analytical applications. Sepimostat (FUT-187 free base) exhibits neuroprotective activity via NR2B N-methyl-D-aspartate receptor antagonism at the Ifenprodil-binding site of the NR2B subunit. Sepimostat inhibits the Ifenprodil binding with a Ki value of 27.7 μM.
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ZIP(Scrambled)
0 ImagesCat. No.: HY-P1391CAS No.: 908012-18-0ZIP(Scrambled) is a scrambled control peptide for zeta inhibitory peptide (ZIP).
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NMDAR antagonist 4
0 ImagesCat. No.: HY-107705CAS No.: 132623-44-0NMDAR antagonist 4 (Compound 8) is the antagonist for NMDA receptor that binds NMDA receptor on glycine site with Ki >100 μM.
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LY 235959
0 ImagesCat. No.: HY-101353CAS No.: 137433-06-8Synonyms: (-)-LY 235959LY 235959 is a competitive N-methyl-D-aspartate (NMDA)-receptor antagonist. LY 235959 potentiates the anticonvulsant action of antiepileptics.
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LY339434
0 ImagesCat. No.: HY-114550CAS No.: 219566-62-8LY339434 is a potent and selective agonist for the hydrochloride receptor GluR5. LY339434 affects the rapid death of neurons through n-methyl-D-aspartate (NMDA) receptors.
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Nelonemdaz (Standard)
0 ImagesCat. No.: HY-106408RCAS No.: 640290-67-1Synonyms: Salfaprodil free base (Standard); Neu2000 (Standard)Nelonemdaz (Standard) is the analytical standard of Nelonemdaz (HY-106408). This product is intended for research and analytical applications. Nelonemdaz (Salfaprodil free base) is an NR2B-selective and uncompetitive antagonist of N-methyl-D-aspartate (NMDA). Nelonemdaz is also a free radical scavenger. Nelonemdaz has excellent neuroprotection against NMDA- and free radical-induced cell death.
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Quinolinic acid-13C7
0 ImagesCat. No.: HY-100807S1CAS No.: 1346642-91-8Quinolinic acid-13C7 is the 13C labeled Quinolinic acid (HY-100807). Quinolinic acid, an endogenous metabolite of tryptophan, is a N-methyl-D-aspartate receptor (NMDA receptor) agonist. Quinolinic acid increases glutamate efflux, induces the generation of ROS, activates nitric oxide synthase, produces excessive NO, leading to calcium ion influx and neuronal apoptosis.
