1. GPCR/G Protein
    Neuronal Signaling
  2. CGRP Receptor

Ubrogepant (Synonyms: MK-1602)

Cat. No.: HY-12366
Handling Instructions

Ubrogepant (MK-1602) is a novel oral calcitonin gene-related peptide receptor (CGRP) antagonist in development for acute treatment of migraine[1].

For research use only. We do not sell to patients.

Ubrogepant Chemical Structure

Ubrogepant Chemical Structure

CAS No. : 1374248-77-7

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  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

Ubrogepant (MK-1602) is a novel oral calcitonin gene-related peptide receptor (CGRP) antagonist in development for acute treatment of migraine[1].

IC50 & Target

MK-1602[1]

Clinical Trial
Solvent & Solubility
In Vitro: 

10 mM in DMSO

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.8197 mL 9.0985 mL 18.1970 mL
5 mM 0.3639 mL 1.8197 mL 3.6394 mL
10 mM 0.1820 mL 0.9099 mL 1.8197 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

549.54

Formula

C₂₉H₂₆F₃N₅O₃

CAS No.

1374248-77-7

SMILES

O=C(C1=CN=C2C(C[[email protected]@]3(C4=CC=CN=C4NC3=O)C2)=C1)N[[email protected]@H]5C(N(CC(F)(F)F)[[email protected]](C)[[email protected]](C6=CC=CC=C6)C5)=O

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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This equation is commonly abbreviated as: C1V1 = C2V2

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× = ×
C1   V1   C2   V2

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Product Name:
Ubrogepant
Cat. No.:
HY-12366
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Ubrogepant

Cat. No.: HY-12366