1. Metabolic Enzyme/Protease
  2. RAR/RXR
  3. AC-261066

AC-261066 

Cat. No.: HY-108532
Handling Instructions

AC-261066 is a potent, orally available and isoform-selective retinoic acid beta2 (RARbeta2) receptor agonist, with a pEC50 of 8.0.

For research use only. We do not sell to patients.

AC-261066 Chemical Structure

AC-261066 Chemical Structure

CAS No. : 870773-76-5

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Description

AC-261066 is a potent, orally available and isoform-selective retinoic acid beta2 (RARbeta2) receptor agonist, with a pEC50 of 8.0[1].

IC50 & Target

RARβ2

8.0 (pEC50)

In Vitro

AC-261066 exhibits good oral bioavailability in rats (F oral = 52%)[1].

Molecular Weight

353.41

Formula

C₁₇H₂₀FNO₄S

CAS No.

870773-76-5

SMILES

O=C(O)C1=CC=C(C2=NC(OCCOCCCC)=C(C)S2)C=C1F

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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Keywords:

AC-261066AC261066AC 261066RAR/RXRRetinoic acid receptorsRetinoid X receptorsisoform-selectiveRARbeta2Inhibitorinhibitorinhibit

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AC-261066
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