BMS-210285
BMS-210285 is a highly selective agonist for the 3 receptor. BMS-210285 has a Ki of 9 nM at the human 3-adrenoceptor. BMS-210285 possesses a 3 intrinsic activity of 83% relative to isoproterenol. BMS-210285 can be studied for obesity and type 2 diabetes research.
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- CAS. Nr.: 344607-69-8
- Formel: C24H25ClF2N2O5S
- Molecular Weight:526.98
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
Chemical Information
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CAS. Nr. 344607-69-8
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Molecular Weight 526.98
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Formel C24H25ClF2N2O5S
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SMILES
CS(=O)(NC1=CC([C@@H](O)CN[C@@H](C2=CC=C(OC(F)F)C=C2)CC3=CC=CC(Cl)=C3)=CC=C1O)=O
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
[1]. Hu, B., & Jennings, L. L. (2003). Orally bioavailable beta 3-adrenergic receptor agonists as potential therapeutic agents for obesity and type-II diabetes. Progress in medicinal chemistry, 41, 167-194. [Content Brief]
[2]. Kordik, C. P., & Reitz, A. B. (1999). Pharmacological treatment of obesity: therapeutic strategies. Journal of medicinal chemistry, 42(2), 181-201. [Content Brief]
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)