LUF5437
LUF5437 is a potent and selective adenosine A1 receptor antagonist with a rat Ki of 7.3 nM. LUF5437 can be used for research on cardiovascular and neurological diseases.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- CAS. Nr.: 331472-34-5
- Formel: C15H11N3O2S
- Molecular Weight:297.33
-
Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Alle Adenosine Receptor Isoform-spezifische Produkte anzeigen
More
Biologische Aktivität
Beschreibung
IC50 & Target
[1]|
rA1 7.3 nM (Ki) |
rA2A 0.57 μM (Ki) |
hA3 0.13 μM (Ki) |
In Vitro
LUF5437 (Compound 8h) acts as a potent and selective adenosine A1 receptor antagonist, with a Ki of 7.3 nM at rat adenosine A1 receptors[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
-
CAS. Nr. 331472-34-5
-
Molecular Weight 297.33
-
Formel C15H11N3O2S
-
SMILES
O=C(NC1=NC(C2=CC=CC=C2)=NS1)C3=CC=C(O)C=C3
-
Versand
Room temperature in continental US; may vary elsewhere.
-
Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)