Azepexole hydrochloride

(Synonyms: B-HT 933 hydrochloride; Oxazoloazepin hydrochloride)
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Azepexole hydrochloride (B-HT 933 dihydrochloride; Oxazoloazepin dihydrochloride) is a selective agonist for α 2-adrenoceptor, with pKi of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively. Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions with IC50 of 78.72 nM. Azepexole hydrochloride exhibits antitussive and analgesic efficacy.

For research use only. We do not sell to patients.

  • Purity: 99.89%
  • CAS No.: 147663-20-5
  • Formula: C9H16ClN3O
  • Molecular Weight:217.70
  • Storage:

    4°C, sealed storage, away from moisture

    * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

  • Biological Activity
  • Chemical Information
  • Purity & Documentation
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All Adrenergic Receptor Isoforms

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