Beloxepin
Based on 1 Customer Validation
Beloxepin (Org 4428) is an orally active synaptosomal noradrenalin reuptake inhibitor and a 5-HT2 receptor antagonist. Beloxepin shows about 100-fold less affine for other monoamine carriers. Beloxepin has antidepressant and pain-relieving effects.
For research use only. We do not sell to patients.
- Purity: 98.04%
- CAS No.: 135928-30-2
- Formula: C19H21NO2
- Molecular Weight:295.38
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Storage:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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5-HT2 Receptor |
Chemical Information
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CAS No. 135928-30-2
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Appearance Solid
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Molecular Weight 295.38
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Formula C19H21NO2
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Color White to off-white
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SMILES
O[C@@]12[C@@](CN(CC2)C)([H])C3=CC=CC(C)=C3OC4=CC=CC=C41
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Synonyms
Org 4428; ADL 6906
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
Purity & Documentation
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Data Sheet (277 KB)
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SDS (557 KB)
- English - EN (557 KB)
- Français - FR (557 KB)
- Deutsch - DE (557 KB)
- Norwegian - NO (557 KB)
- Español - ES (557 KB)
- Swedish - SV (557 KB)
- Italian - IT (557 KB)
- Korean - KR (557 KB)
- Portuguese - PT (557 KB)
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Handling Instructions (2659 KB)
References
[1]. Lorenzo Di Cesare Mannelli, et al. α2 Adrenoceptor: a Target for Neuropathic Pain Treatment. Mini Rev Med Chem. 2017;17(2):95-107. [Content Brief]
[2]. Craig T Hartrick. Noradrenergic reuptake inhibition in the treatment of pain. Expert Opin Investig Drugs. 2012 Dec;21(12):1827-34. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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