S1427
S1427 is a tranylcypromine-derived LSD1 inhibitor with the IC50 of 390 nM and Ki of 80 nM. S1427 exhibits desirable hERG channel inhibition and microsomal stability profiles. Inhibition of LSD1 partially reduces the proliferation of cancer cells.
Nos produits utilisent uniquement pour la recherche. Nous ne vendons pas aux patients.
- CAS No.: 2447061-40-5
- Formule: C25H29F3N4O2
- Masse moléculaire:474.52
-
Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
|
KDM1/LSD1 |
Chemical Information
-
CAS No. 2447061-40-5
-
Masse moléculaire 474.52
-
Formule C25H29F3N4O2
-
SMILES
O=C(N1CCC2(CC1)CCNC2)CN[C@H]3C[C@@H]3C4=C(C(F)=CC(F)=C4)OCC5=CC=CN=C5F
-
Livraison
Room temperature in continental US; may vary elsewhere.
-
Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)