Clomiphene-d5 citrate
Clomiphene-d5 (citrate) is the deuterium labeled Enclomiphene citrate. Enclomiphene citrate is a potent and orally active oestrogen receptor antagonist, with antioestrogenic property.
For research use only. We do not sell to patients.
- CAS No.: 1217200-17-3
- Formula: C32H31D5ClNO8
- Molecular Weight:603.11
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
1. This compound can be used as a tracer
2. This compound can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.
Chemical Information
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CAS No. 1217200-17-3
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Unlabeled Cas 50-41-9
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Molecular Weight 603.11
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Formula C32H31D5ClNO8
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SMILES
C(CC(O)=O)(CC(O)=O)(C(O)=O)O.C(=C(Cl)C1=CC=CC=C1)(C2=CC=C(OCCN(CC)CC)C=C2)C3=C(C(=C(C(=C3[2H])[2H])[2H])[2H])[2H]
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Synonyms
Clomifene-d5 citrate; (Z/E)-Enclomiphene-d5 citrate; (Z/E)-Enclomifene-d5 citrate
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
[1]. Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216. [Content Brief]
[2]. Fontenot GK, et al. Differential effects of isomers of clomiphene citrate on reproductive tissues in male mice. BJU Int. 2016 Feb;117(2):344-50. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Clomiphene-d5 citrate Related Classifications
HY-118861AS1 Related Classifications
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