CVT-5440
CVT-5440 is a xanthine based, selective, high affinity A2B adenosine receptors (AdoR) antagonist with a Ki of 50 nM (selectivity A1> 200; A2A>200; A3>167). CVT-5440 has the potential for asthma research.
For research use only. We do not sell to patients.
- CAS No.: 531506-64-6
- Formula: C27H28N6O5
- Molecular Weight:516.55
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Adenosine Receptor Isoforms
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Biological Activity
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A2B 50 nM (Ki) |
A1 >10,000 nM (Ki) |
A2A >5,000 nM (Ki) |
Chemical Information
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CAS No. 531506-64-6
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Molecular Weight 516.55
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Formula C27H28N6O5
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SMILES
O=C(N1CCC)N(CCC)C2=C(N=C(C3=CC=C(OCC4=NOC(C5=CC=CC(OC)=C5)=N4)C=C3)N2)C1=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)