1. GPCR/G Protein
    Neuronal Signaling
  2. Opioid Receptor
  3. CYT-1010

CYT-1010 

Cat. No.: HY-123534 Purity: 99.74%
Handling Instructions

CYT-1010 is a mu-opioid receptor agonist extracted from patent WO2013173730A2, with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively.

For research use only. We do not sell to patients.

CYT-1010 Chemical Structure

CYT-1010 Chemical Structure

CAS No. : 213769-33-6

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 481 In-stock
Estimated Time of Arrival: December 31
5 mg USD 350 In-stock
Estimated Time of Arrival: December 31
10 mg USD 550 In-stock
Estimated Time of Arrival: December 31
50 mg USD 1650 In-stock
Estimated Time of Arrival: December 31
100 mg   Get quote  
200 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

Based on 1 publication(s) in Google Scholar

Other Forms of CYT-1010:

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Description

CYT-1010 is a mu-opioid receptor agonist extracted from patent WO2013173730A2, with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively[1].

IC50 & Target

EC50: 13.1 nM (beta-arrestin), 0.0053 nM (cAMP)[1]

Molecular Weight

624.73

Formula

C₃₅H₄₀N₆O₅

CAS No.

213769-33-6

SMILES

OC1=CC=C(C=C1)C[[email protected]@H](C(N[[email protected]](CCCCNC2=O)C(N[[email protected]@H](CC3=CNC4=C3C=CC=C4)C(N[[email protected]]2CC5=CC=CC=C5)=O)=O)=O)N

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 125 mg/mL (200.09 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.6007 mL 8.0035 mL 16.0069 mL
5 mM 0.3201 mL 1.6007 mL 3.2014 mL
10 mM 0.1601 mL 0.8003 mL 1.6007 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.08 mg/mL (3.33 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.08 mg/mL (3.33 mM); Clear solution

*All of the co-solvents are provided by MCE.
References
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Keywords:

CYT-1010CYT1010CYT 1010Opioid ReceptorInhibitorinhibitorinhibit

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Product name:
CYT-1010
Cat. No.:
HY-123534
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