E-2508 free base

E-2508 free base is an orally active and highly selective corticotropin-releasing factor type 1 receptor (CRF1) antagonist with anxiolytic effects (Ki=11 nM). E-2508 free base blocks CRF-induced cAMP accumulation via CRF1 receptor inhibition. E-2508 free base is promising for research of stress-related psychiatric disorders, such as anxiety and depression.

For research use only. We do not sell to patients.

  • CAS No.: 685885-75-0
  • Formula: C29H39N3O4
  • Molecular Weight:493.64
  • Storage:

    Please store the product under the recommended conditions in the Certificate of Analysis.

  • Biological Activity
  • Chemical Information
  • Purity & Documentation
  • References
  • Help & FAQs

All CRFR Isoforms

More
100 mg

Get Quote In-stock

Please select quantity
Amount: USD 0.00