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  2. ELA-21 (human)

ELA-21 (human) 

Cat. No.: HY-P2249
Handling Instructions

ELA-21 (human) is an apelin receptor agonist with a pKi of 8.52. ELA-21 (human) completely inhibits Forskolin-induced cAMP production and stimulates β-arrestin recruitment with subnanomolar potencies. ELA-21 (human) is an agonist in G-protein-dependent and -independent pathways.

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ELA-21 (human) Chemical Structure

ELA-21 (human) Chemical Structure

CAS No. : 2245073-05-4

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Description

ELA-21 (human) is an apelin receptor agonist with a pKi of 8.52. ELA-21 (human) completely inhibits Forskolin-induced cAMP production and stimulates β-arrestin recruitment with subnanomolar potencies. ELA-21 (human) is an agonist in G-protein-dependent and -independent pathways[1].

Molecular Weight

2587.14

Formula

C₁₁₂H₁₈₄N₄₀O₂₅S₃

CAS No.

2245073-05-4

Sequence

Leu-Arg-Lys-His-Asn-Cys-Leu-Gln-Arg-Arg-Cys-Met-Pro-Leu-His-Ser-Arg-Val-Pro-Phe-Pro (Disulfide bridge: Cys6-Cys11)

Sequence Shortening

LRKHNCLQRRCMPLHSRVPFP (Disulfide bridge: Cys6-Cys11)

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

ELA-21 (human)OthersApelinG-proteincAMPβ-arrestinInhibitorinhibitorinhibit

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