Enpp-1-IN-21
Based on 1 Customer Validation
Enpp-1-IN-21 (compound 4g) is an inhibitor of ecto-nucleotide pyrophosphatase/phosphodiesterase 1 (ENPP1), with IC50 values for ENPP1 and ENPP3 at 0.45 and 0.19 μM, respectively.
For research use only. We do not sell to patients.
- Purity: 99.07%
- CAS No.: 2803505-78-2
- Formula: C21H16F3NO5S
- Molecular Weight:451.42
-
Storage:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
Biological Activity
Chemical Information
-
CAS No. 2803505-78-2
-
Appearance Solid
-
Molecular Weight 451.42
-
Formula C21H16F3NO5S
-
Color White to light yellow
-
SMILES
O=C(C1=CC=C(C)C=C1)NC2=CC=C(C=C2)OS(=O)(C3=CC=C(C=C3)OC(F)(F)F)=O
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
DMSO : 100 mg/mL (221.52 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
-
Data Sheet (266 KB)
-
SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
-
Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.2152 mL | 11.0762 mL | 22.1523 mL | 55.3808 mL |
| 5 mM | 0.4430 mL | 2.2152 mL | 4.4305 mL | 11.0762 mL | |
| 10 mM | 0.2215 mL | 1.1076 mL | 2.2152 mL | 5.5381 mL | |
| 15 mM | 0.1477 mL | 0.7384 mL | 1.4768 mL | 3.6921 mL | |
| 20 mM | 0.1108 mL | 0.5538 mL | 1.1076 mL | 2.7690 mL | |
| 25 mM | 0.0886 mL | 0.4430 mL | 0.8861 mL | 2.2152 mL | |
| 30 mM | 0.0738 mL | 0.3692 mL | 0.7384 mL | 1.8460 mL | |
| 40 mM | 0.0554 mL | 0.2769 mL | 0.5538 mL | 1.3845 mL | |
| 50 mM | 0.0443 mL | 0.2215 mL | 0.4430 mL | 1.1076 mL | |
| 60 mM | 0.0369 mL | 0.1846 mL | 0.3692 mL | 0.9230 mL | |
| 80 mM | 0.0277 mL | 0.1385 mL | 0.2769 mL | 0.6923 mL | |
| 100 mM | 0.0222 mL | 0.1108 mL | 0.2215 mL | 0.5538 mL |