EP4 receptor agonist 2
Based on 1 Customer Validation
EP4 receptor agonist 2 (compound 31) a potent EP4 receptor agonist with an EC50 value of 0.8 nM; Ki values of >100000, 38000, 3.1 nM for EP2, EP3, EP4 respectively.
The product specifications provided below refer solely to the active content of EP4 receptor agonist 2.
For research use only. We do not sell to patients.
- Purity : 99.20%
- CAS No.: 493035-81-7
- Formula: C27H32ClNO4
- Molecular Weight:470.00
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Storage:
Solution, -20°C, 2 years
Biological Activity
Description
The product specifications provided below refer solely to the active content of EP4 receptor agonist 2.
IC50 & Target
[1]|
EP4 0.8 nM (EC50) |
EP2 >100000 nM (Ki) |
EP3 38000 nM (Ki) |
EP4 3.1 nM (Ki) |
Cellular Effect
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| CHO | EC50 |
0.8 nM
Compound: 31
|
Agonist activity against recombinant prostanoid EP4 receptor stably transfected in CHO cells
Agonist activity against recombinant prostanoid EP4 receptor stably transfected in CHO cells
|
[PMID: 15026044] |
Chemical Information
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CAS No. 493035-81-7
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Appearance Liquid
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Molecular Weight 470.00
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Formula C27H32ClNO4
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Color Colorless to light yellow
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SMILES
CC1=C(C=CC(Cl)=C1)C2=CC(C(O)/C=C/[C@@H]3N(C(CC3)=O)CCCCCCC(O)=O)=CC=C2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Solution, -20°C, 2 years
Purity & Documentation
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Data Sheet (287 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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Handling Instructions (2659 KB)
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)