EP4 receptor agonist 2
Based on 1 Customer Validation
EP4 receptor agonist 2 (compound 31) a potent EP4 receptor agonist with an EC50 value of 0.8 nM; Ki values of >100000, 38000, 3.1 nM for EP2, EP3, EP4 respectively.
For research use only. We do not sell to patients.
- Purity: 99.0%
- CAS No.: 493035-81-7
- Formula: C27H32ClNO4
- Molecular Weight:470.00
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Storage:
Solution, -20°C, 2 years
Biological Activity
|
EP4 0.8 nM (EC50) |
EP2 >100000 nM (Ki) |
EP3 38000 nM (Ki) |
EP4 3.1 nM (Ki) |
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| CHO | EC50 |
0.8 nM
Compound: 31
|
Agonist activity against recombinant prostanoid EP4 receptor stably transfected in CHO cells
Agonist activity against recombinant prostanoid EP4 receptor stably transfected in CHO cells
|
[PMID: 15026044] |
Chemical Information
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CAS No. 493035-81-7
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Appearance Liquid
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Molecular Weight 470.00
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Formula C27H32ClNO4
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Color Colorless to light yellow
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SMILES
CC1=C(C=CC(Cl)=C1)C2=CC(C(O)/C=C/[C@@H]3N(C(CC3)=O)CCCCCCC(O)=O)=CC=C2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Solution, -20°C, 2 years
Purity & Documentation
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Data Sheet (272 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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Handling Instructions (2659 KB)
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)