ER degrader 9
ER degrader 9 is a bifunctional estrogen receptor degrader that mediates ER protein degradation in MCF7 cells.
For research use only. We do not sell to patients.
- CAS No.: 3023359-75-0
- Formula: C40H48N4O2
- Molecular Weight:616.83
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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ER |
ER degrader 9 (Compound 1) mediates ER protein degradation in MCF7 cells. According to the ER protein degradation assay, its DC50 is < 10 nM, and 50 % < Dmax < 65 %[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 3023359-75-0
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Molecular Weight 616.83
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Formula C40H48N4O2
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SMILES
CC(C)(/C=C(C(N1CCN(CC1)CC2CCN(CC2)C3=CC=C(C=C3)[C@H]4[C@H](CCC5=CC(O)=CC=C54)C6=CC=CC=C6)=O)/C#N)C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)