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United States

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Referencia número: HY-113683

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AZ 12488024

(Synonyms: AZD7268)

AZ 12488024 (AZD7268) is a SNC80 (HY-101202) derivative and a δ-opioid receptor agonist. AZ 12488024 is available for research into major depressive disorder.

Para uso exclusivo en investigación. No vendemos a pacientes.

No. CAS: 1018988-00-5
Fòrmula: C₂₉H₃₀N₄O₂S
Peso molecular:498.64

Almacenamiento:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (265 KB)

AZ 12488024 Chemical Structure

No. CAS: 1018988-00-5

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Actividad biológica
- Descripciòn
- Cellular Effect
- Ensayo clínico
Chemical Information
Pureza y Documentación
Referencias
Calculators
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Bioz

Actividad biológica

Descripciòn

AZ 12488024 (AZD7268) is a SNC80 (HY-101202) derivative and a δ-opioid receptor agonist. AZ 12488024 is available for research into major depressive disorder^[1].

Ver todos los productos específicos de isoformas Opioid Receptor :

Cellular Effect

Cell Line	Type	Value	Description	References
HEK293	IC₅₀	0.28 nM Compound: 20	Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranes Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranes	[PMID: 22197137]
HEK293	IC₅₀	460 nM Compound: 20	Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranes Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranes	[PMID: 22197137]

Ensayo clínico

NCT Number	Sponsor	Condition	Start Date	Phase A549
NCT01329991	Plexxikon\|		2011-05	PHASE1

Chemical Information

No. CAS 1018988-00-5
Peso molecular 498.64
Fòrmula C₂₉H₃₀N₄O₂S
SMILES

O=C(C1=CC=C(C=C1)/C(C2=C3N=CC=CC3=CC=C2)=C4CCN(CC\4)CC5=CSC=N5)N(C)CCO
Synonyms

AZD7268
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureza y Documentación

Select Batch:

Pureza: 99.98%

Assay: 99.98%

ee.: 99.98%

Ficha de datos (265 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instrucciones de manejo (2659 KB)

Referencias

[1]. Fujii H, et al. Non-peptidic δ opioid receptor agonists and antagonists (2000–2012)[J]. Expert Opinion on Therapeutic Patents, 2013, 23(9): 1181-1208. [Content Brief]

Calculators

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Actividad biológica
- Descripciòn
- Ensayo clínico
Chemical Information
Pureza y Documentación
Referencias

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AZ 12488024

Ver todos los productos específicos de isoformas Opioid Receptor

Actividad biológica

Chemical Information

Pureza y Documentación

Referencias

Calculators

Help & FAQs

AZ 12488024 Related Classifications

HY-113683 Related Classifications