LUF5437
LUF5437 is a potent and selective adenosine A1 receptor antagonist with a rat Ki of 7.3 nM. LUF5437 can be used for research on cardiovascular and neurological diseases.
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- No. CAS: 331472-34-5
- Fòrmula: C15H11N3O2S
- Peso molecular:297.33
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Ver todos los productos específicos de isoformas Adenosine Receptor
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Actividad biológica
Descripciòn
IC50 & Target
[1]|
rA1 7.3 nM (Ki) |
rA2A 0.57 μM (Ki) |
hA3 0.13 μM (Ki) |
In Vitro
LUF5437 (Compound 8h) acts as a potent and selective adenosine A1 receptor antagonist, with a Ki of 7.3 nM at rat adenosine A1 receptors[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 331472-34-5
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Peso molecular 297.33
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Fòrmula C15H11N3O2S
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SMILES
O=C(NC1=NC(C2=CC=CC=C2)=NS1)C3=CC=C(O)C=C3
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)