Org 25543
Org 25543 is a selective inhibitor of the glycine transporter 2, exhibiting analgesic properties in a rat model of chronic pain.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 363628-88-0
- Fòrmula: C24H32N2O4
- Peso molecular:412.52
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| CHO | IC50 |
16 nM
Compound: 35; ORG-25543
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Inhibition of human GlyT2 stably expressed in CHO cells assessed as reduction in [3H]glycine uptake incubated for 10 mins by liquid scintillation counting method
Inhibition of human GlyT2 stably expressed in CHO cells assessed as reduction in [3H]glycine uptake incubated for 10 mins by liquid scintillation counting method
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[PMID: 31774679] |
Chemical Information
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No. CAS 363628-88-0
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Peso molecular 412.52
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Fòrmula C24H32N2O4
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SMILES
COC(C=C(C(NCC1(CCCC1)N(C)C)=O)C=C2OC)=C2OCC3=CC=CC=C3
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Org 25543 Related Classifications
HY-107527A Related Classifications
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