GDI2-IN-1
GDI2-IN-1 (compound (+)-37) is a GDP-dissociation inhibitor beta (GDI2) inhibitor with an IC50 of 2.87 μM and a KD of 36 μM. GDI2-IN-1 exhibits excellent in vivo antitumor activity in GDI2-overexpressing pancreatic xenograft models.
For research use only. We do not sell to patients.
- Formula: C42H47FN4O3
- Molecular Weight:674.85
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Chemical Information
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Molecular Weight 674.85
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Formula C42H47FN4O3
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SMILES
O[C@](C[C@@H]1C)(CC2=CN(CC3=CC=C(F)C=C3)N=N2)C[C@@]4([H])N1CCC5=C4C=C(OCC6=CC(C)=CC(C)=C6)C(OCC7=CC(C)=CC(C)=C7)=C5
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)