1. GPCR/G Protein
  2. Free Fatty Acid Receptor
  3. GPR40 agonist 5

GPR40 agonist 5 

Cat. No.: HY-147678
Handling Instructions

GPR40 agonist 5 (compound I-14) is an orally active and potent GPR40 (G protein coupled receptor 40) agonist, with an EC50 of 47 nM. GPR40 agonist 5 decreases the levels of blood glucose and improves the glucose tolerance. GPR40 agonist 5 has sufficient effectiveness for the control of hyperglycemia state in type 2 diabetic mice.

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GPR40 agonist 5 Chemical Structure

GPR40 agonist 5 Chemical Structure

CAS No. : 2443384-60-7

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Description

GPR40 agonist 5 (compound I-14) is an orally active and potent GPR40 (G protein coupled receptor 40) agonist, with an EC50 of 47 nM. GPR40 agonist 5 decreases the levels of blood glucose and improves the glucose tolerance. GPR40 agonist 5 has sufficient effectiveness for the control of hyperglycemia state in type 2 diabetic mice[1].

IC50 & Target

EC50: 47 ± 9.8 nM (GPR40)[1]

Molecular Weight

440.49

Formula

C27H24N2O4

CAS No.
SMILES

CC#CC(C1=CC=C(C=C1)OCC2=CN3C=C(N=C3C=C2)C4=CC=C(C=C4)OC)CC(O)=O

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Please store the product under the recommended conditions in the Certificate of Analysis.

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Product Name:
GPR40 agonist 5
Cat. No.:
HY-147678
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