YM-254891
YM-254891 is a YM-254890 (HY-111557) analogue and Gαq/11 inhibitor. YM-254891 can be isolated from the fermentation broth of Chromobacterium sp. QS3666. YM-254891 inhibits ADP-induced platelet aggregation.
For research use only. We do not sell to patients.
- CAS No.: 726188-99-4
- Formula: C47H71N7O15
- Molecular Weight:974.10
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Biological Activity
-
Chemical Information
- Purity & Documentation
- References
-
Help & FAQs
Biological Activity
|
Microbial Metabolite |
YM-254891 inhibits 2MeSADP-induced Ca2+ influx in P2Y1-C6-15 cells with an IC50 of 0.23 μM[1].
YM-254891 inhibits ADP-induced platelet aggregation in platelet-rich plasma with an IC50 of 0.27 μM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
-
CAS No. 726188-99-4
-
Molecular Weight 974.10
-
Formula C47H71N7O15
-
SMILES
CCC(N[C@@H]([C@H](O)C(C)C)C(O[C@@H]([C@@]1([H])C(N([C@@](C(O[C@@H]([C@@H](C(O[C@@H](C(N(C(C(N[C@H](C(N([C@H](C(N1)=O)C)C)=O)C)=O)=C)C)=O)CC2=CC=CC=C2)=O)NC(C)=O)C)=O)([H])[C@@H](C)OC)C)=O)C(C)C)=O)=O
-
Structure Classification
-
Initial Source
Chromobacterium sp
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
YM-254891 Related Classifications
HY-N17826 Related Classifications
Powered by Bioz