Pridinol
Pridinol is an orally active, blood-brain permeable, muscarinic acetylcholine receptor (mAChR)-directed muscle relaxant. Pridinol reduces the conduction of impulses to spinal motor neurons and exerts muscle relaxant activity. Pridinol inhibits skeletal muscle contractures in diseases of both central and peripheral origin and can be used in research in the field of musculoskeletal diseases.
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研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 511-45-5
- 分子式: C20H25NO
- 分子量:295.42
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
生物活性
The in vitro dissolution characteristics of Pridinol are slightly affected by pH (pH 1.2, 4.5, 6.8)[1].
The lower limit of detection of Pridinol in biological samples is 0.0500 ng/mL and the upper limit is 50 ng/mL[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 511-45-5
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分子量 295.42
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分子式 C20H25NO
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SMILES
OC(C1=CC=CC=C1)(C2=CC=CC=C2)CCN3CCCCC3
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
[1]. Richter M, et al. Pharmacokinetics of oral pridinol: Results of a randomized, crossover bioequivalence trial in healthy subjects. Int J Clin Pharmacol Ther. 2021 Jun;59(6):471-477. [Content Brief]
[2]. Lauricella L, et al. Effectiveness rehabilitative therapy and Pridinol Mesylate in low back pain. Front Med (Lausanne) . 2025 Jan 22;11:1470996. [Content Brief]
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)