Epigenetic Reader Domain Control
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trans-BAY-850
0 ImagesCat. No.: HY-119254APurity: 99.30%
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(R)-INCB054329
0 Images(R)-INCB054329 is the isomer of INCB054329 (HY-112504), and can be used as an experimental control. INCB054329 is a potent BET inhibitor.
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GSK 525768A
0 ImagesGSK 525768A is the inactive enantiomer of GSK525762A. GSK 525768A has no activity towards BET.
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(R)-I-BET762 carboxylic acid
0 ImagesSynonyms: (R)-Molibresib carboxylic acid; (R)-GSK525762A carboxylic acid; (R)-PROTAC BRD4-binding moiety 2(R)-I-BET762 carboxylic acid, the R-enantiomer of I-BET762 carboxylic acid (HY-107443). I-BET762 carboxylic acid is an I-BET762-based warhead ligand for conjugation reactions of PROTAC targeting on BET. I-BET762 carboxylic acid is a BRD4 inhibitor with a pIC50 value of 5.1.
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D-Moses
0 ImagesCat. No.: HY-101125BCAS No.: 2084850-77-9Synonyms: D-45
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(2R,3R)-GSK973
0 ImagesCat. No.: HY-138563A(2R,3R)-GSK973 is an isomer of GSK973. GSK973 is a highly selective, orally bioavailable inhibitor of the BD2s (second bromodomains) of the BET family.
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cis-SIM1
0 ImagesCat. No.: HY-141438ACAS No.: 2719051-98-4cis-SIM1 is a negative control of SIM1.
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Mivebresib-alkyne
0 ImagesCat. No.: HY-169980CAS No.: 2409674-37-7Mivebresib-alkyne (Compound 25), a Mivebresib (HY-100015) derivative, can be used for BRD4 targeted PROTAC synthesis through click reaction.
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(R)-I-BET762 carboxylic acid (Standard)
0 ImagesSynonyms: (R)-Molibresib carboxylic acid (Standard); (R)-GSK525762A carboxylic acid (Standard); (R)-PROTAC BRD4-binding moiety 2 (Standard)(R)-I-BET762 carboxylic acid (Standard) is the analytical standard of (R)-I-BET762 carboxylic acid (HY-107443A). This product is intended for research and analytical applications. (R)-I-BET762 carboxylic acid, the R-enantiomer of I-BET762 carboxylic acid (HY-107443). I-BET762 carboxylic acid is an I-BET762-based warhead ligand for conjugation reactions of PROTAC targeting on BET. I-BET762 carboxylic acid is a BRD4 inhibitor with a pIC50 value of 5.1.
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