1. PROTAC
  2. Ligand for Target Protein
  3. PROTAC BRD4-binding moiety 2

PROTAC BRD4-binding moiety 2 

Cat. No.: HY-107443 Purity: 96.04% ee.: 99.52%
Handling Instructions

PROTAC BRD4-binding moiety 2 is a BRD4(1) inhibitor with an IC50 of 7.9 μM.

For research use only. We do not sell to patients.

PROTAC BRD4-binding moiety 2 Chemical Structure

PROTAC BRD4-binding moiety 2 Chemical Structure

CAS No. : 1300019-38-8

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 288 In-stock
Estimated Time of Arrival: December 31
1 mg USD 110 In-stock
Estimated Time of Arrival: December 31
5 mg USD 330 In-stock
Estimated Time of Arrival: December 31
10 mg USD 550 In-stock
Estimated Time of Arrival: December 31
50 mg USD 1650 In-stock
Estimated Time of Arrival: December 31
100 mg   Get quote  
200 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

Other Forms of PROTAC BRD4-binding moiety 2:

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Description

PROTAC BRD4-binding moiety 2 is a BRD4(1) inhibitor with an IC50 of 7.9 μM.

IC50 & Target

BRD4(1)

7.9 μM (IC50)

In Vitro

PROTAC BRD4-binding moiety 2 (compound 32) is a BRD4 (1) inhibitor with an IC50 of 7.9 μM[1].

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 7.14 mg/mL (17.99 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.5200 mL 12.5999 mL 25.1997 mL
5 mM 0.5040 mL 2.5200 mL 5.0399 mL
10 mM 0.2520 mL 1.2600 mL 2.5200 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

396.83

Formula

C₂₀H₁₇ClN₄O₃

CAS No.

1300019-38-8

SMILES

CC1=NN=C2[[email protected]](CC(O)=O)N=C(C3=CC=C(Cl)C=C3)C4=C(C=CC(OC)=C4)N21

Shipping

Room temperature in continental US; may vary elsewhere

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
PROTAC BRD4-binding moiety 2
Cat. No.:
HY-107443
Quantity:

PROTAC BRD4-binding moiety 2

Cat. No.: HY-107443