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(E,E)-GLL398

(E,E)-GLL398 is a selective estrogen receptor degrader with potent binding activity to ERα (IC50 = 1.14 nM). (E,E)-GLL398 can effectively degrade ERα in MCF-7 breast cancer cells (IC50 = 0.21 μM). The introduced boronic acid group of (E,E)-GLL398 gives it superior oral bioavailability, with an AUC of 36.9 μg·h/mL in rats, which is significantly higher than that of GW7604.

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  • CAS No.: 2077980-83-5
  • 화학식: C25H23BO4
  • 분자량:398.26
  • 보관:

    Please store the product under the recommended conditions in the Certificate of Analysis.

  • (E,E)-GLL398 Chemical Structure
    (E,E)-GLL398 Chemical Structure
CAS No.: 2077980-83-5
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All Estrogen Receptor/ERR Isoforms

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    (E,E)-GLL398 Chemical Structure
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  • (E,E)-GLL398