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Cat. No.: HY-123447

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GR-175737

GR 175737 is a partial histamine H3 receptor agonist, with an EC₅₀ of 7.8 nM. GR 175737 can be used in the research of inflammatory diseases.

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CAS No.: 176860-26-7
화학식: C₁₄H₁₃ClN₄O
분자량:288.73

보관:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (266 KB)

GR-175737 Chemical Structure

CAS No.: 176860-26-7

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- 제품 설명
- IC₅₀ & Target
Chemical Information
순도&문서
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

제품 설명

GR 175737 is a partial histamine H3 receptor agonist, with an EC₅₀ of 7.8 nM. GR 175737 can be used in the research of inflammatory diseases^[1].

IC₅₀ & Target^[1]

H₃ receptor

7.8 nM (EC₅₀)

All Histamine Receptor Isoforms :

Chemical Information

CAS No. 176860-26-7
분자량 288.73
화학식 C₁₄H₁₃ClN₄O
SMILES

ClC1=CC=C(C=C1)CC2=NOC(CCC3=CN=CN3)=N2
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.

순도&문서

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (266 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Soudijn W, et al. Structure–activity relationships of inverse agonists for G‐protein‐coupled receptors. Medicinal research reviews, 2005, 25(4): 398-426.

Calculators

몰농도 계산기

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

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Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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MOQ

Minimum order quantity

100 mg

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Amount: USD 0.00

Biological Activity
- 제품 설명
- IC₅₀ & Target
Chemical Information
순도&문서
References

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GR-175737

All Histamine Receptor Isoforms

Biological Activity

Chemical Information

순도&문서

References

Calculators

Help & FAQs

GR-175737 Related Classifications

HY-123447 Related Classifications