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Cat. No.: HY-124912

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VUF-6884

VUF-6884 (Compound 7j) is a histamine receptor (Histamine Receptor) ligand with activity toward human H4R and H1R. Its pEC₅₀ and pK_i values against human H4R are 7.70 and 7.55, respectively, while those against human H1R are 8.17 and 8.11, respectively. VUF-6884 competitively binds to the orthosteric binding site of human H4R to displace histamine, and exhibits inverse agonist activity at human H1R.

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CAS No.: 3455-10-5
화학식: C₁₈H₁₈ClN₃O
분자량:327.81

보관:

Please store the product under the recommended conditions in the Certificate of Analysis.

VUF-6884 Chemical Structure

CAS No.: 3455-10-5

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

제품 설명

All Histamine Receptor Isoforms :

Chemical Information

CAS No. 3455-10-5
분자량 327.81
화학식 C₁₈H₁₈ClN₃O
SMILES

ClC1=CC=C2N=C(C=3C=CC=CC3OC2=C1)N4CCN(C)CC4
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.

순도&문서

Handling Instructions (2659 KB)

References

[1]. Smits RA, et al. Characterization of the histamine H4 receptor binding site. Part 1. Synthesis and pharmacological evaluation of dibenzodiazepine derivatives. J Med Chem. 2006;49(15):4512-4516. [Content Brief]

Calculators

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biological Activity
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Chemical Information
순도&문서
References

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VUF-6884

All Histamine Receptor Isoforms

Biological Activity

Chemical Information

순도&문서

References

Calculators

Help & FAQs

VUF-6884 Related Classifications

HY-124912 Related Classifications