2. GPCR/G Protein
    Neuronal Signaling
  3. Neuropeptide Y Receptor
  4. M617 TFA

M617 TFA 

Cat. No.: HY-P1131A Purity: 99.91%
COA Handling Instructions

M617 TFA is a selective galanin receptor 1 (GAL1) agonist, with Kis of 0.23 and 5.71 nM for GAL1 and GAL2, respectively. M617 TFA, acting through its central GAL1, can promote GLUT4 expression and enhance GLUT4 content in the cardiac muscle of type 2 diabetic rats.

For research use only. We do not sell to patients.

Custom Peptide Synthesis

M617 TFA Chemical Structure

M617 TFA Chemical Structure

Size Price Stock Quantity
5 mg USD 365 In-stock
Estimated Time of Arrival: December 31
10 mg USD 620 In-stock
Estimated Time of Arrival: December 31
50 mg   Get quote  
100 mg   Get quote  

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Based on 1 publication(s) in Google Scholar

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Description

M617 TFA is a selective galanin receptor 1 (GAL1) agonist, with Kis of 0.23 and 5.71 nM for GAL1 and GAL2, respectively. M617 TFA, acting through its central GAL1, can promote GLUT4 expression and enhance GLUT4 content in the cardiac muscle of type 2 diabetic rats[1][2].

Molecular Weight

2475.67

Appearance

Solid

Formula

C114H162F3N29O30
Sequence

Gly-Trp-Thr-Leu-Asn-Ser-Ala-Gly-Tyr-Leu-Leu-Gly-Pro-Gln-Pro-Pro-Gly-Phe-Ser-Pro-NH2
Sequence Shortening

GWTLNSAGYLLGPQPPGFSPFR-NH2
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Sealed storage, away from moisture and light

Powder -80°C 2 years
-20°C 1 year

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
Solvent & Solubility
In Vitro: 

H2O : 33.33 mg/mL (13.46 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 0.4039 mL 2.0197 mL 4.0393 mL
5 mM 0.0808 mL 0.4039 mL 0.8079 mL
10 mM 0.0404 mL 0.2020 mL 0.4039 mL
*Please refer to the solubility information to select the appropriate solvent.
Purity & Documentation
References
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

M617M 617M-617Neuropeptide Y ReceptorNPY receptorGLUT4type2diabeticanti-nociceptioncardiovascularInhibitorinhibitorinhibit

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M617 TFA
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