1. Neuronal Signaling
  2. Beta-secretase
  3. OM99-2 TFA

OM99-2 TFA 

Cat. No.: HY-P2713A
Handling Instructions

OM99-2 TFA, an eight residue peptidomimetic, tight-binding inhibitor of human brain memapsin 2 with a Ki value of 9.58 nM. OM99-2 TFA is significantly advanced the development of BACE1 inhibitor, has the potential for the research of the Alzheimer's disease.

For research use only. We do not sell to patients.

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OM99-2 TFA Chemical Structure

OM99-2 TFA Chemical Structure

CAS No. : 2504147-81-1

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Description

OM99-2 TFA, an eight residue peptidomimetic, tight-binding inhibitor of human brain memapsin 2 with a Ki value of 9.58 nM[1]. OM99-2 TFA is significantly advanced the development of BACE1 inhibitor[2], has the potential for the research of the Alzheimer's disease[3].

IC50 & Target

Ki: 9.58 nM (memapsin 2)

In Vitro

Memapsin 2 (BACE) is an aspartyl protease known as beta-secretase that acts on the production of the beta-amyloid peptide in the human brain[4].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

1007.02

Formula

C₄₃H₆₅F₃N₈O₁₆

CAS No.
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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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OM99-2 TFA
Cat. No.:
HY-P2713A
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